From a collaboration of Schools and Departments at University of Michigan, Ann Arbor MI (US), discovery of a highly potent and effective proteolysis targeting chimeras ER degrader.
AUTHORS: Jiantao Hu, Biao Hu, Mingliang Wang, Fuming Xu, Bukeyan Miao, Chao-Yie Yang, Mi Wang, Zhaomin Liu, Daniel F. Hayes, Krishnapriya Chinnaswamy, James Delproposto, Jeanne Stuckey, and Shaomeng Wang
SOURCE: J. Med. Chem., DOI: 10.1021/acs.jmedchem.8b01572 - Publication Date (Web): January 18, 2019
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